HQ005 is a Molecular glue degrader of cyclin K (DC50 = 41 nM). Reference: Lv, L., Chen, P., Cao, L., Li, Y., Zeng, Z., Cui, Y., Wu, Q., Li, J., Wang, J.-H., Dong, M.-Q., Qi, X.,Han, T., Discovery of a molecular glue promoting CDK12-DDB1 interaction to trigger cyclin K degradation. eLife 2020, 9, e59994.
Product Name |
HQ005 |
Synonyms |
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CAS Number |
2750644-31-4 |
Related CAS |
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Molecular Formula |
C15H15N5O2S2 |
Molecular Weight |
361.44 |
SMILES |
CC1=CN=C(NC(=O)CC2=CSC(NC3=NC(CO)=CC=C3)=N2)S1 |
Purity (HPLC) |
98% |
Shipping Conditions |
Room Temperature |
Storage Conditions |
Refrigerated |
Regulatory Statemen: |
For Research Use Only |