TMX-4113 is a degrader of phosphodiesterase 6D (PDE6D) and casein kinase 1a(CK1a). TMX-4113 can be used for the research of cancer. Reference: Teng, M., Lu, W., Donovan, K. A., Sun, J., Krupnick, N. M., Nowak, R. P., Li, Y.-D., Sperling, A. S., Zhang, T., Ebert, B. L., Fischer, E. S.,Gray, N. S., Development of PDE6D and CK1a Degraders through Chemical Derivatization of FPFT-2216. Journal of Medicinal Chemistry 2022, 65, 747-756.
Product Name |
TMX-4113 |
Synonyms |
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CAS Number |
2766385-92-4 |
Related CAS |
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Molecular Formula |
C12H12N4O2S2 |
Molecular Weight |
308.37 |
SMILES |
CSC1=CSC=C1C1=CN(N=N1)C1CCC(=O)NC1=O |
Purity (HPLC) |
98% |
Shipping Conditions |
Room Temperature |
Storage Conditions |
Refrigerated |
Regulatory Statemen: |
For Research Use Only |